Press Release

G-Protein Coupled Receptors Market to Grow with a CAGR of 5.23% through 2030

Increasing investment in precision medicine and the growing adoption of AI-driven drug development for GPCR-targeted therapies, is expected to drive the Global G-Protein Coupled Receptors Market growth in the forecast period, 2026-2030

 

According to TechSci Research report, “G-Protein Coupled Receptors Market – Global Industry Size, Share, Trends, Competition Forecast & Opportunities, 2030F”, the Global G-Protein Coupled Receptors Market stood at USD 3.95 Billion in 2024 and is expected to reach USD 5.37 Billion by 2030 with a CAGR of 5.23% during the forecast period. The Global G-Protein Coupled Receptors (GPCR) Market is experiencing rapid expansion due to its vital role in cellular signaling and drug development. GPCRs are among the most versatile drug targets, regulating numerous physiological functions such as immune response, neurotransmission, and hormone regulation. With pharmaceutical companies focusing on next-generation therapeutics, GPCR-targeted drugs are gaining traction in treating diseases like diabetes, psychiatric disorders, and autoimmune conditions. Advances in structural elucidation techniques, including X-ray crystallography and nuclear magnetic resonance (NMR) spectroscopy, have significantly improved the understanding of GPCR mechanisms, fostering drug discovery. The emergence of selective GPCR modulators and combination therapies has expanded treatment options, further propelling market growth.

The increasing demand for innovative treatment options is fueling investments in GPCR-targeted biologics and peptide-based drugs. The rise of precision pharmacology has enabled the development of GPCR allosteric modulators, offering better receptor selectivity and reduced side effects. The adoption of artificial intelligence (AI) in GPCR modeling has streamlined ligand-binding studies, expediting drug discovery pipelines. Growing interest in functional selectivity has led to the identification of biased agonists, allowing for more targeted therapeutic effects. Expansion in gene-editing technologies such as CRISPR is facilitating research into GPCR gene regulation, unlocking new possibilities for disease modification. The integration of lab-on-a-chip technologies for high-throughput GPCR screening has also enhanced drug testing efficiency, accelerating market development.

The emergence of GPCR-targeted therapies in immuno-oncology presents a major growth avenue, with researchers exploring novel GPCR-mediated pathways for cancer treatment. The expansion of biosimilar and biologic drugs targeting GPCRs is expected to create cost-effective treatment alternatives, enhancing patient access. Increasing research into orphan GPCRs, which currently lack identified ligands, holds potential for discovering breakthrough therapies. The integration of nanotechnology in GPCR drug delivery is improving therapeutic precision, reducing systemic side effects. Partnerships between biotech firms and academic institutions are fostering innovation, leading to a deeper understanding of GPCR pharmacology and expanding the range of druggable GPCR targets. With continued technological advancements and industry

 

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The Global G-Protein Coupled Receptors Market is segmented into product, assay type, application, regional distribution, and company.

Based on the Application, Inflammation Research emerged as the fastest growing segment in the Global G-Protein Coupled Receptors Market during the forecast period. This is due to the increasing recognition of GPCRs as key regulators of immune and inflammatory responses. GPCRs play a crucial role in mediating signal transduction in various inflammatory pathways, making them attractive targets for drug development. The rising prevalence of chronic inflammatory diseases, including rheumatoid arthritis, inflammatory bowel disease, and psoriasis, has driven extensive research into GPCR-targeted therapies. Pharmaceutical and biotechnology companies are actively investing in identifying novel GPCR modulators that can help regulate immune responses, reduce inflammation, and provide more effective treatment options. Recent advancements in high-throughput screening technologies have facilitated the identification of GPCR-based drug candidates, accelerating the development of new anti-inflammatory drugs. The growing demand for biologics and small-molecule drugs targeting GPCRs in inflammation-related disorders is further fueling market expansion. Additionally, regulatory approvals for GPCR-targeted therapies in inflammation management are encouraging further research and innovation in this domain. The increasing burden of inflammatory diseases, coupled with continuous advancements in GPCR drug discovery and development, is expected to drive significant growth in this segment during the forecast period.

Based on the Region, Asia-Pacific emerged as the fastest growing region in the Global G-Protein Coupled Receptors Market during the forecast period. This is due to increasing investments in drug discovery, rising healthcare expenditures, and expanding pharmaceutical and biotechnology industries. The region is experiencing rapid advancements in biomedical research, supported by government initiatives and funding for innovative drug development. Countries such as China, Japan, and India are becoming key hubs for GPCR-targeted research due to the availability of skilled researchers, improved research infrastructure, and collaborations between academic institutions and pharmaceutical companies. Pharmaceutical companies are focusing on developing novel GPCR-based drugs to address the growing disease burden. Furthermore, the presence of a large patient population and evolving regulatory frameworks supporting faster drug approvals have encouraged market expansion. The growth of contract research organizations (CROs) and increased foreign direct investment in the region are further propelling the adoption of GPCR research technologies. With continuous advancements in drug discovery, increasing clinical trials, and a strong pipeline of GPCR-targeted therapeutics, Asia-Pacific is expected to witness significant market growth during the forecast period.

 

Major companies operating in Global G-Protein Coupled Receptors Market are:

  • Thermo Fisher Scientific Inc.
  • PerkinElmer Inc.
  • Promega Corporation
  • Merck KGaA
  • Abcam plc
  • Becton, Dickinson and Company
  • Danaher Corporation
  • QIAGEN N.V.
  • Bio-Techne Corporation
  • WuXi AppTec

 

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The Global G-Protein Coupled Receptors Market is expanding due to the increasing adoption of advanced drug screening technologies that enhance the efficiency and accuracy of GPCR-targeted drug discovery. The integration of artificial intelligence (AI) and machine learning (ML) in the research and development of GPCR-based therapies is helping to predict molecular interactions, optimize drug design, and identify novel therapeutic targets. These technologies enable faster and more cost-effective discovery processes, increasing the number of GPCR-targeted drug candidates entering clinical trials. The growing emphasis on AI-driven drug discovery platforms is driving innovations and accelerating the development of new GPCR-targeted treatments.,” said Mr. Karan Chechi, Research Director of TechSci Research, a research-based management consulting firm.

 

G-Protein Coupled Receptors Market - Global Industry Size, Share, Trends, Opportunity, and Forecast, Segmented By Product (Cell Lines, Detection Kits, Cell Culture Reagents, Ligands), By Assay Type (cAMP Functional Assays, Calcium Functional Assays, β-Arrestin Functional Assays, Radioligand Binding & GTPγS Functional Assays, Internalization Assays, Trafficking Assays, Others), By Application (Cancer Research, CNS Research, Metabolic Research, Cardiovascular Research, Respiratory Research, Inflammation Research, Others), By Region and Competition, 2020-2030F”, has evaluated the future growth potential of Global G-Protein Coupled Receptors Market and provides statistics & information on market size, structure and future market growth. The report intends to provide cutting-edge market intelligence and help decision makers take sound investment decisions. Besides, the report also identifies and analyzes the emerging trends along with essential drivers, challenges, and opportunities in Global G-Protein Coupled Receptors Market.

 

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